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Synthesis and Functional Characterization of Substituted Isoquinolinones as MT(2)-Selective Melatoninergic Ligands
A series of substituted isoquinolinones were synthesized and their binding affinities and functional activities towards human melatonin MT(1) and MT(2) receptors were evaluated. Structure-activity relationship analysis revealed that substituted isoquinolinones bearing a 3-methoxybenzyloxyl group at...
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| Pubblicato in: | PLoS One |
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| Autori principali: | , , , , |
| Natura: | Artigo |
| Lingua: | Inglês |
| Pubblicazione: |
Public Library of Science
2014
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| Soggetti: | |
| Accesso online: | https://ncbi.nlm.nih.gov/pmc/articles/PMC4257560/ https://ncbi.nlm.nih.gov/pubmed/25479338 https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1371/journal.pone.0113638 |
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