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Basal and β-adrenergic regulation of the cardiac calcium channel Ca(V)1.2 requires phosphorylation of serine 1700

L-type calcium (Ca(2+)) currents conducted by voltage-gated Ca(2+) channel Ca(V)1.2 initiate excitation–contraction coupling in cardiomyocytes. Upon activation of β-adrenergic receptors, phosphorylation of Ca(V)1.2 channels by cAMP-dependent protein kinase (PKA) increases channel activity, thereby a...

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Pubblicato in:Proc Natl Acad Sci U S A
Autori principali: Fu, Ying, Westenbroek, Ruth E., Scheuer, Todd, Catterall, William A.
Natura: Artigo
Lingua:Inglês
Pubblicazione: National Academy of Sciences 2014
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC4246329/
https://ncbi.nlm.nih.gov/pubmed/25368181
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1073/pnas.1419129111
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