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Thiourea-Catalyzed Enantioselective Addition of Indoles to Pyrones: Alkaloid Cores with Quaternary Carbons

[Image: see text] We report the development of a catalytic method for the enantioselective addition of indoles to pyrone-derived electrophiles. Arylpyrrolidino-derived thioureas catalyze the addition with high stereoselectivity in the presence of catalytic quantities of an achiral Brønsted acid. The...

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Bibliographic Details
Published in:J Am Chem Soc
Main Authors: Yeung, Charles S., Ziegler, Robert E., Porco, John A., Jacobsen, Eric N.
Format: Artigo
Language:Inglês
Published: American Chemical Society 2014
Online Access:https://ncbi.nlm.nih.gov/pmc/articles/PMC4235369/
https://ncbi.nlm.nih.gov/pubmed/25213353
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/ja508523g
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