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Picomolar Inhibitors of HIV-1 Reverse Transcriptase: Design and Crystallography of Naphthyl Phenyl Ethers

[Image: see text] Catechol diethers that incorporate a 6-cyano-1-naphthyl substituent have been explored as non-nucleoside inhibitors of HIV-1 reverse transcriptase (NNRTIs). Promising compounds are reported that show midpicomolar activity against the wild-type virus and sub-20 nM activity against v...

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Detalles Bibliográficos
Publicado en:ACS Med Chem Lett
Main Authors: Lee, Won-Gil, Frey, Kathleen M., Gallardo-Macias, Ricardo, Spasov, Krasimir A., Bollini, Mariela, Anderson, Karen S., Jorgensen, William L.
Formato: Artigo
Idioma:Inglês
Publicado: American Chemical Society 2014
Acceso en liña:https://ncbi.nlm.nih.gov/pmc/articles/PMC4233359/
https://ncbi.nlm.nih.gov/pubmed/25408842
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/ml5003713
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