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Preparation, Physicochemical Characterization and In-vitro Dissolution Studies of Diosmin-cyclodextrin Inclusion Complexes

Diosmin, a vascular-protecting agent, is practically insoluble in water, and its oral absorption is limited by its extremely low dissolution rate. In this study, β-cyclodextrin (βCD) and 2-hydroxypropyl-β-cyclodextrin (HPβCD) were obtained to improve the solubility and dissolution rate of diosmin. P...

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Publicat a:Iran J Pharm Res
Autors principals: Ai, Fengwei, Ma, Yingli, Wang, Jiayu, Li, Yanfeng
Format: Artigo
Idioma:Inglês
Publicat: Shaheed Beheshti University of Medical Sciences 2014
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Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC4232776/
https://ncbi.nlm.nih.gov/pubmed/25587299
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