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Drug Target Identification Using a Trypanosome Overexpression Library

Elucidation of molecular targets is very important for lead optimization during the drug development process. We describe a direct method to find targets of antitrypanosomal compounds against Trypanosoma brucei using a trypanosome overexpression library. As proof of concept, we treated the library w...

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Autors principals: Begolo, Daniela, Erben, Esteban, Clayton, Christine
Format: Artigo
Idioma:Inglês
Publicat: American Society for Microbiology 2014
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Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC4187942/
https://ncbi.nlm.nih.gov/pubmed/25049244
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1128/AAC.03338-14
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