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Incorporating target-mediated drug disposition in a minimal physiologically-based pharmacokinetic model for monoclonal antibodies

Target-mediated drug disposition (TMDD) usually accounts for nonlinear pharmacokinetics (PK) of drugs whose distribution and/or clearance are affected by their targets owing to high affinity and limited capacity. TMDD is frequently reported for monoclonal antibodies (mAb) for such reason. Minimal ph...

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Autors principals: Cao, Yanguang, Jusko, William J.
Format: Artigo
Idioma:Inglês
Publicat: 2014
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC4167346/
https://ncbi.nlm.nih.gov/pubmed/25077917
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1007/s10928-014-9372-2
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