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Probing Biased/Partial Agonism at the G Protein-Coupled A(2B) Adenosine Receptor()

G protein-coupled A(2B) adenosine receptor (AR) regulates numerous important physiological functions, but its activation by diverse A(2B)AR agonists is poorly profiled. We probed potential partial and/or biased agonism in cell lines expressing variable levels of endogenous or recombinant A(2B)AR. In...

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Wedi'i Gadw mewn:
Manylion Llyfryddiaeth
Prif Awduron: Gao, Zhan-Guo, Balasubramanian, Ramachandran, Kiselev, Evgeny, Wei, Qiang, Jacobson, Kenneth A.
Fformat: Artigo
Iaith:Inglês
Cyhoeddwyd: 2014
Pynciau:
Mynediad Ar-lein:https://ncbi.nlm.nih.gov/pmc/articles/PMC4128710/
https://ncbi.nlm.nih.gov/pubmed/24853985
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bcp.2014.05.008
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