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Activation of p53 signaling by MI-63 induces apoptosis in acute myelogenous leukemia cells

Non-mutational inactivation of p53 is frequent in acute myeloid leukemia (AML) via overexpression of MDM2. We report that treatment with MI-63, a novel inhibitor of MDM2, activates p53 signaling to induce apoptosis in AML cell lines and primary samples. Cell lines naturally devoid of p53 or expressi...

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Detalhes bibliográficos
Main Authors: Samudio, Ismael J, Duvvuri, Seshagiri, Clise-Dwyer, Karen, Watt, Julie C, Mak, Duncan, Kantarjian, Hagop, Yang, Dajun, Ruvolo, Vivian, Borthakur, Gautam
Formato: Artigo
Idioma:Inglês
Publicado em: 2010
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Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC4122268/
https://ncbi.nlm.nih.gov/pubmed/20423286
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3109/10428191003731325
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