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A gatekeeper residue for NEDD8 activating enzyme inhibition by MLN4924

Inhibition of NEDD8 activating enzyme (NAE) has emerged as a highly promising approach to treat cancer through the adenosine sulfamate analogue MLN4924. Here we show that selective pressure results in HCT116 colorectal carcinoma cells with decreased MLN4924 sensitivity and identify a single nucleoti...

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Autori principali: Toth, Julia I., Yang, Li, Dahl, Russell, Petroski, Matthew D.
Natura: Artigo
Lingua:Inglês
Pubblicazione: 2012
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC4120840/
https://ncbi.nlm.nih.gov/pubmed/22832224
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.celrep.2012.02.006
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