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Advances in the discovery of N-acylethanolamine acid amidase inhibitors

N-acylethanolamine acid amidase (NAAA) is a cysteine amidase that hydrolyzes saturated or monounsaturated fatty acid ethanolamides, such as palmitoylethanolamide (PEA) and oleoylethanolamide (OEA). PEA has been shown to exert analgesic and anti-inflammatory effects by engaging peroxisome proliferato...

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Main Authors: Bandiera, Tiziano, Ponzano, Stefano, Piomelli, Daniele
Formato: Artigo
Idioma:Inglês
Publicado: 2014
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Acceso en liña:https://ncbi.nlm.nih.gov/pmc/articles/PMC4117721/
https://ncbi.nlm.nih.gov/pubmed/24798679
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.phrs.2014.04.011
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