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Selective PPARγ modulator INT131 normalizes insulin signaling defects and improves bone mass in diet-induced obese mice

INT131 is a potent non-thiazolidinedione (TZD)-selective peroxisome proliferator-activated receptor-γ modulator being developed for the treatment of type 2 diabetes. In preclinical studies and a phase II clinical trial, INT131 has been shown to lower glucose levels and ameliorate insulin resistance...

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Bibliografske podrobnosti
Main Authors: Lee, Dae Ho, Huang, Hu, Choi, Kangduk, Mantzoros, Christos, Kim, Young-Bum
Format: Artigo
Jezik:Inglês
Izdano: American Physiological Society 2012
Teme:
Online dostop:https://ncbi.nlm.nih.gov/pmc/articles/PMC4116349/
https://ncbi.nlm.nih.gov/pubmed/22215652
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1152/ajpendo.00569.2011
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