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Selective Inhibition of Bacterial Topoisomerase I by alkynyl-bisbenzimidazoles

Hoechst dyes are well known DNA binders that non-selectively inhibit the function of mammalian topoisomerase I and II. Herein, we show that Hoechst 33258 based bisbenzimidazoles (DPA 151–154), containing a terminal alkyne, are effective and selective inhibitors of E. coli. topoisomerase I. These bis...

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Detalhes bibliográficos
Main Authors: Ranjan, Nihar, Fulcrand, Geraldine, King, Ada, Brown, Joseph, Jiang, Xiuping, Leng, Fenfei, Arya, Dev P.
Formato: Artigo
Idioma:Inglês
Publicado em: 2014
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC4112416/
https://ncbi.nlm.nih.gov/pubmed/25083189
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1039/C4MD00140K
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