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Rational design and validation of a Tip60 histone acetyltransferase inhibitor

Histone acetylation is required for many aspects of gene regulation, genome maintenance and metabolism and dysfunctional acetylation is implicated in numerous diseases, including cancer. Acetylation is regulated by histone acetyltransferases (HATs) and histone deacetylases and currently, few general...

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Detalhes bibliográficos
Main Authors: Gao, Chunxia, Bourke, Emer, Scobie, Martin, Famme, Melina Arcos, Koolmeister, Tobias, Helleday, Thomas, Eriksson, Leif A., Lowndes, Noel F., Brown, James A. L.
Formato: Artigo
Idioma:Inglês
Publicado em: Nature Publishing Group 2014
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC4064327/
https://ncbi.nlm.nih.gov/pubmed/24947938
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/srep05372
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