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METOCLOPRAMIDE IS METABOLIZED BY CYP2D6 AND IS A REVERSIBLE INHIBITOR, BUT NOT INACTIVATOR, OF CYP2D6

1. Metoclopramide is a widely used clinical drug in a variety of medical settings with rare acute dystonic events reported. The aim of this study was to assess a previous report of inactivation of CYP2D6 by metoclopramide, to determine the contribution of various CYPs to metoclopramide metabolism, a...

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Autors principals: Livezey, Mara R., Briggs, Erran D., Bolles, Amanda K., Nagy, Leslie D., Fujiwara, Rina, Furge, Laura Lowe
Format: Artigo
Idioma:Inglês
Publicat: 2013
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC4059401/
https://ncbi.nlm.nih.gov/pubmed/24010633
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3109/00498254.2013.835885
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