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The Rhodadyns, a New Class of Small Molecule Inhibitors of Dynamin GTPase Activity

[Image: see text] Six focused rhodanine-based libraries, 60 compounds in total, were synthesized and evaluated as potential dynamin I GTPase inhibitors. Twenty-six were more potent than the lead compound with 13 returning IC(50) values ≤10 μM, making the Rhodadyn series among the most active dynamin...

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Autori principali: Robertson, Mark J., Hadzic, Gordana, Ambrus, Joseph, Pomè, D. Yuri, Hyde, Emily, Whiting, Ainslie, Mariana, Anna, von Kleist, Lisa, Chau, Ngoc, Haucke, Volker, Robinson, Phillip J., McCluskey, Adam
Natura: Artigo
Lingua:Inglês
Pubblicazione: American Chemical Society 2012
Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC4025782/
https://ncbi.nlm.nih.gov/pubmed/24900478
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/ml200284s
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