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Targeting the c-Kit Promoter G-quadruplexes with 6-Substituted Indenoisoquinolines

[Image: see text] Herein, we demonstrate the design, synthesis, biophysical properties, and preliminary biological evaluation of 6-substituted indenoisoquinolines as a new class of G-quadruplex stabilizing small molecule ligands. We have synthesized 6-substituted indenoisoquinolines 1a−e in two step...

Ausführliche Beschreibung

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Bibliographische Detailangaben
Hauptverfasser: Bejugam, Mallesham, Gunaratnam, Mekala, Müller, Sebastian, Sanders, Deborah A., Sewitz, Sven, Fletcher, Jonathan A., Neidle, Stephen, Balasubramanian, Shankar
Format: Artigo
Sprache:Inglês
Veröffentlicht: American Chemical Society 2010
Online Zugang:https://ncbi.nlm.nih.gov/pmc/articles/PMC4017300/
https://ncbi.nlm.nih.gov/pubmed/24900212
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/ml100062z
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