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Rapid Delivery of Diazepam from Supersaturated Solutions Prepared Using Prodrug/Enzyme Mixtures: Toward Intranasal Treatment of Seizure Emergencies

Current treatments for seizure emergencies, such as status epilepticus, include intravenous or rectal administration of benzodiazepines. While intranasal delivery of these drugs is desirable, the small volume of the nasal cavity and low drug solubility pose significant difficulties. Here, we prepare...

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Autori principali: Kapoor, Mamta, Winter, Tate, Lis, Lev, Georg, Gunda I., Siegel, Ronald A.
Natura: Artigo
Lingua:Inglês
Pubblicazione: Springer US 2014
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC4012037/
https://ncbi.nlm.nih.gov/pubmed/24700272
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1208/s12248-014-9596-5
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