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Novel 16-substituted bifunctional derivatives of huperzine B: multifunctional cholinesterase inhibitors

AIM: To design novel bifunctional derivatives of huperzine B (HupB) based on the concept of dual binding site of acetylcholinesterase (AChE) and evaluate their pharmacological activities for seeking new drug candidates against Alzheimer's disease (AD). METHODS: Novel 16-substituted bifunctional...

पूर्ण विवरण

में बचाया:
ग्रंथसूची विवरण
मुख्य लेखकों: Shi, Yu-fang, Zhang, Hai-yan, Wang, Wei, Fu, Yan, Xia, Yu, Tang, Xi-can, Bai, Dong-lu, He, Xu-chang
स्वरूप: Artigo
भाषा:Inglês
प्रकाशित: Nature Publishing Group 2009
विषय:
ऑनलाइन पहुंच:https://ncbi.nlm.nih.gov/pmc/articles/PMC4006674/
https://ncbi.nlm.nih.gov/pubmed/19578388
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/aps.2009.91
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