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Inhibition of mutant BRAF splice variant signaling by next generation, selective RAF inhibitors

Vemurafenib and dabrafenib block MEK-ERK1/2 signaling and cause tumor regression in the majority of advanced-stage BRAF(V600E) melanoma patients; however, acquired resistance and paradoxical signaling have driven efforts for more potent and selective RAF inhibitors. Next generation RAF inhibitors, s...

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Bibliografiske detaljer
Main Authors: Basile, Kevin J., Le, Kaitlyn, Hartsough, Edward J., Aplin, Andrew E.
Format: Artigo
Sprog:Inglês
Udgivet: 2014
Fag:
Online adgang:https://ncbi.nlm.nih.gov/pmc/articles/PMC3988223/
https://ncbi.nlm.nih.gov/pubmed/24422853
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1111/pcmr.12218
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