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Simplified Cyclic Analogs of Bastadin-5. Structure Activity Relationships for Modulation of the RyR1/FKBP12 Ca(2+) Channel Complex

Bastadin-5, a brominated macro-dilactam from the marine sponge Ianthella basta, enhances release of Ca(2+) from stores within the sarcoplasmic reticulum (SR) of muscle and non-muscle cells by modulating RyR1/FKBP12 complex. Analogs of bastadin-5 present desirable targets for SAR studies to shed ligh...

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Detalles Bibliográficos
Main Authors: Masuno, Makoto N., Pessah, Isaac N., Olmstead, Marilyn M., Molinski, Tadeusz F.
Formato: Artigo
Idioma:Inglês
Publicado: 2006
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Acceso en liña:https://ncbi.nlm.nih.gov/pmc/articles/PMC3987770/
https://ncbi.nlm.nih.gov/pubmed/16854055
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/jm050708u
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