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Investigation of Chalcones as Selective Inhibitors of the Breast Cancer Resistance Protein: Critical Role of Methoxylation in both Inhibition Potency and Cytotoxicity

[Image: see text] ABCG2 plays a major role in anticancer-drug efflux and related tumor multidrug resistance. Potent and selective ABCG2 inhibitors with low cytotoxicity were investigated among a series of 44 chalcones and analogues (1,3-diarylpropenones), by evaluating their inhibitory effect on the...

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Bibliografski detalji
Glavni autori: Valdameri, Glaucio, Gauthier, Charlotte, Terreux, Raphaël, Kachadourian, Rémy, Day, Brian J., Winnischofer, Sheila M. B., Rocha, Maria E. M., Frachet, Véronique, Ronot, Xavier, Di Pietro, Attilio, Boumendjel, Ahcène
Format: Artigo
Jezik:Inglês
Izdano: 2012
Teme:
Online pristup:https://ncbi.nlm.nih.gov/pmc/articles/PMC3983950/
https://ncbi.nlm.nih.gov/pubmed/22449016
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/jm2016528
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