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Amphiphilic drug interactions with model cellular membranes are influenced by lipid chain-melting temperature

Small-molecule amphiphilic species such as many drug molecules frequently exhibit low-to-negligible aqueous solubility, and generally have no identified transport proteins assisting their distribution, yet are able to rapidly penetrate significant distances into patient tissue and even cross the blo...

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Autors principals: Casey, Duncan, Charalambous, Kalypso, Gee, Antony, Law, Robert V., Ces, Oscar
Format: Artigo
Idioma:Inglês
Publicat: The Royal Society 2014
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Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC3973356/
https://ncbi.nlm.nih.gov/pubmed/24621813
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1098/rsif.2013.1062
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