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Selective Allosteric Enhancement of Agonist Binding and Function at Human A(3) Adenosine Receptors by a Series of Imidazoquinoline Derivatives

We have identified a series of 1H-imidazo-[4,5-c]quinolines as selective allosteric enhancers of human A(3) adenosine receptors. Several of these compounds potentiated both the potency and maximal efficacy of agonist-induced responses and selectively decreased the dissociation of the agonist N(6)-(4...

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書誌詳細
主要な著者: Gao, Zhan-Guo, Kim, Seong Gon, Soltysiak, Kelly A., Melman, Neli, Ijzerman, Adriaan P., Jacobson, Kenneth A.
フォーマット: Artigo
言語:Inglês
出版事項: 2002
主題:
オンライン・アクセス:https://ncbi.nlm.nih.gov/pmc/articles/PMC3953617/
https://ncbi.nlm.nih.gov/pubmed/12065758
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