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TTT-3002 is a novel FLT3 tyrosine kinase inhibitor with activity against FLT3-associated leukemias in vitro and in vivo

More than 35% of acute myeloid leukemia (AML) patients harbor a constitutively activating mutation in FMS-like tyrosine kinase-3 (FLT3). The most common type, internal tandem duplication (ITD), confers poor prognosis. We report for the first time on TTT-3002, a tyrosine kinase inhibitor (TKI) that i...

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Autori principali: Ma, Hayley, Nguyen, Bao, Li, Li, Greenblatt, Sarah, Williams, Allen, Zhao, Ming, Levis, Mark, Rudek, Michelle, Duffield, Amy, Small, Donald
Natura: Artigo
Lingua:Inglês
Pubblicazione: American Society of Hematology 2014
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC3945863/
https://ncbi.nlm.nih.gov/pubmed/24408321
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1182/blood-2013-08-523035
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