Chargement en cours...

Effect of anchoring 4-anilidopiperidines to opioid peptides

We report here the design, synthesis, and in vitro characterization of new opioid peptides featuring a 4-anilidopiperidine moiety. Despite the fact that the chemical structures of fentanyl surrogates have been found suboptimal per se for the opioid activity, the corresponding conjugates with opioid...

Description complète

Enregistré dans:
Détails bibliographiques
Auteurs principaux: Petrov, Ravil R., Lee, Yeon Sun, Vardanyan, Ruben S., Liu, Lu, Ma, Shou-wu, Davis, Peg, Lai, Josephine, Porreca, Frank, Vanderah, Todd W., Hruby, Victor J.
Format: Artigo
Langue:Inglês
Publié: 2013
Sujets:
Accès en ligne:https://ncbi.nlm.nih.gov/pmc/articles/PMC3942532/
https://ncbi.nlm.nih.gov/pubmed/23623418
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bmcl.2013.03.065
Tags: Ajouter un tag
Pas de tags, Soyez le premier à ajouter un tag!