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YM201636, an inhibitor of retroviral budding and PIKfyve-catalyzed PtdIns(3,5)P(2) synthesis, halts glucose entry by insulin in adipocytes

Silencing of PIKfyve, the sole enzyme for PtdIns(3,5)P(2) biosynthesis that controls proper endosome dynamics, inhibits retroviral replication. A novel PIKfyve-specific inhibitor YM201636 disrupts retroviral budding at 800 nM, suggesting its potential use as an antiretroviral therapeutic. Because PI...

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Autori principali: Ikonomov, Ognian C., Sbrissa, Diego, Shisheva, Assia
Natura: Artigo
Lingua:Inglês
Pubblicazione: 2009
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC3910513/
https://ncbi.nlm.nih.gov/pubmed/19289105
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bbrc.2009.03.063
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