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Discovery of new G-quadruplex binding chemotypes

We report here on the discovery and preliminary evaluation of a novel non-macrocyclic low molecular weight quadruplex-stabilizing chemotype. The lead compounds, based on a furan core, show high G-quadruplex stabilisation and selectivity as well as potent in vitro anti-proliferative activity.

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Detalhes bibliográficos
Main Authors: Ohnmacht, Stephan A., Varavipour, Ehsan, Nanjunda, Rupesh, Pazitna, Ingrida, Di Vita, Gloria, Gunaratnam, Mekala, Kumar, Arvind, Ismail, Mohamed A., Boykin, David W., Wilson, W. David, Neidle, Stephen
Formato: Artigo
Idioma:Inglês
Publicado em: 2014
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC3901018/
https://ncbi.nlm.nih.gov/pubmed/24302123
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1039/c3cc48616h
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