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A retro-inverso TAT-like peptide designed to deliver cysteamine to cells

A retro-inverso, TAT-like peptide wherein lysine residues are replaced with cysteine residues bearing a disulfide-linked cysteamine group is found to engage in thiol–disulfide exchange with cysteine. These peptides are transported into cells and localize to lysosomes. Cellular uptake is enhanced in...

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Detalhes bibliográficos
Main Authors: Lim, Jongdoo, Pellois, Jean-Philippe, Simanek, Eric E.
Formato: Artigo
Idioma:Inglês
Publicado em: 2010
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC3881279/
https://ncbi.nlm.nih.gov/pubmed/20843689
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bmcl.2010.07.046
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