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Polypeptide Modulators of TRPV1 Produce Analgesia without Hyperthermia

Transient receptor potential vanilloid 1 receptors (TRPV1) play a significant physiological role. The study of novel TRPV1 agonists and antagonists is essential. Here, we report on the characterization of polypeptide antagonists of TRPV1 based on in vitro and in vivo experiments. We evaluated the ab...

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Hlavní autoři: Andreev, Yaroslav A., Kozlov, Sergey A., Korolkova, Yuliya V., Dyachenko, Igor A., Bondarenko, Dmitrii A., Skobtsov, Denis I., Murashev, Arkadii N., Kotova, Polina D., Rogachevskaja, Olga A., Kabanova, Natalia V., Kolesnikov, Stanislav S., Grishin, Eugene V.
Médium: Artigo
Jazyk:Inglês
Vydáno: MDPI 2013
Témata:
On-line přístup:https://ncbi.nlm.nih.gov/pmc/articles/PMC3877906/
https://ncbi.nlm.nih.gov/pubmed/24351908
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/md11125100
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