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Polypeptide Modulators of TRPV1 Produce Analgesia without Hyperthermia

Transient receptor potential vanilloid 1 receptors (TRPV1) play a significant physiological role. The study of novel TRPV1 agonists and antagonists is essential. Here, we report on the characterization of polypeptide antagonists of TRPV1 based on in vitro and in vivo experiments. We evaluated the ab...

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Bibliografski detalji
Glavni autori: Andreev, Yaroslav A., Kozlov, Sergey A., Korolkova, Yuliya V., Dyachenko, Igor A., Bondarenko, Dmitrii A., Skobtsov, Denis I., Murashev, Arkadii N., Kotova, Polina D., Rogachevskaja, Olga A., Kabanova, Natalia V., Kolesnikov, Stanislav S., Grishin, Eugene V.
Format: Artigo
Jezik:Inglês
Izdano: MDPI 2013
Teme:
Online pristup:https://ncbi.nlm.nih.gov/pmc/articles/PMC3877906/
https://ncbi.nlm.nih.gov/pubmed/24351908
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/md11125100
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