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The Relative Contributions of CYP3A4 and CYP3A5 to the Metabolism of Vinorelbine

Vinorelbine is a semisynthetic vinca alkaloid used in the treatment of advanced breast and non-small cell lung cancers. Vincristine, a related vinca alkaloid, is 9-fold more efficiently metabolized by CYP3A5 than by CYP3A4 in vitro. This study quantified the relative contribution of CYP3A4 and CYP3A...

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Autors principals: Topletz, Ariel R., Dennison, Jennifer B., Barbuch, Robert J., Hadden, Chad E., Hall, Stephen D., Renbarger, Jamie L.
Format: Artigo
Idioma:Inglês
Publicat: The American Society for Pharmacology and Experimental Therapeutics 2013
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Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC3876810/
https://ncbi.nlm.nih.gov/pubmed/23780963
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1124/dmd.113.051094
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