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Two Distinct Allosteric Binding Sites at α4β2 Nicotinic Acetylcholine Receptors Revealed by NS206 and NS9283 Give Unique Insights to Binding Activity-associated Linkage at Cys-loop Receptors

Positive allosteric modulators (PAMs) of α4β2 nicotinic acetylcholine receptors have the potential to improve cognitive function and alleviate pain. However, only a few selective PAMs of α4β2 receptors have been described limiting both pharmacological understanding and drug-discovery efforts. Here,...

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Détails bibliographiques
Auteurs principaux: Olsen, Jeppe A., Kastrup, Jette S., Peters, Dan, Gajhede, Michael, Balle, Thomas, Ahring, Philip K.
Format: Artigo
Langue:Inglês
Publié: American Society for Biochemistry and Molecular Biology 2013
Sujets:
Accès en ligne:https://ncbi.nlm.nih.gov/pmc/articles/PMC3861648/
https://ncbi.nlm.nih.gov/pubmed/24169695
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1074/jbc.M113.498618
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