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Synthesis of 19-substituted geldanamycins with altered conformations and their binding to heat shock protein Hsp90

The benzoquinone ansamycin geldanamycin and its derivatives are inhibitors of heat shock protein Hsp90, an emerging target for novel therapeutic agents both in cancer and in neurodegeneration. However, toxicity of these compounds to normal cells has been ascribed to reaction with thiol nucleophiles...

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Detalhes bibliográficos
Main Authors: Kitson, Russell R. A., Chang, Chuan-Hsin, Xiong, Rui, Williams, Huw E. L., Davis, Adrienne L., Lewis, William, Dehn, Donna L., Siegel, David, Roe, S. Mark, Prodromou, Chrisostomos, Ross, David, Moody, Christopher J.
Formato: Artigo
Idioma:Inglês
Publicado em: 2013
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Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC3839848/
https://ncbi.nlm.nih.gov/pubmed/23511419
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/nchem.1596
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