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Identification of Tamoxifen-Induced Coregulator Interaction Surfaces within the Ligand-Binding Domain of Estrogen Receptors

Tamoxifen is a selective estrogen receptor (ER) modulator that is clinically used as an antagonist to treat estrogen-dependent breast cancers but displays unwanted agonistic effects in other tissues. Previous studies on ERα have delineated a role of the N-terminal activation function AF-1 in mediati...

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Bibliografski detalji
Glavni autori: Heldring, Nina, Nilsson, Maria, Buehrer, Benjamin, Treuter, Eckardt, Gustafsson, Jan-Åke
Format: Artigo
Jezik:Inglês
Izdano: American Society for Microbiology 2004
Teme:
Online pristup:https://ncbi.nlm.nih.gov/pmc/articles/PMC381632/
https://ncbi.nlm.nih.gov/pubmed/15060164
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1128/MCB.24.8.3445-3459.2004
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