Caricamento...

Strategic Combination of DNA-Damaging Agent and PARP Inhibitor Results in Enhanced Cytotoxicity

PARP inhibitors (PARPi) are under clinical trial for combination cancer chemotherapy. In the presence of a PARPi, PARP-1 binds DNA strand breaks but cannot produce poly(ADP-ribose) polymers or undergo auto-poly(ADP-ribosyl)ation. DNA binding is persistent, hindering DNA repair. Methylated bases form...

Descrizione completa

Salvato in:
Dettagli Bibliografici
Autori principali: Horton, Julie K., Wilson, Samuel H.
Natura: Artigo
Lingua:Inglês
Pubblicazione: Frontiers Media S.A. 2013
Soggetti:
Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC3786324/
https://ncbi.nlm.nih.gov/pubmed/24137565
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3389/fonc.2013.00257
Tags: Aggiungi Tag
Nessun Tag, puoi essere il primo ad aggiungerne! !