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N,N-Disubstituted Piperazines: Synthesis and Affinities at α4β2* and α7* Neuronal Nicotinic Acetylcholine Receptors

A series of N,N-disubstituted piperazines were prepared and evaluated for binding to α4β2* and α7* neuronal nicotinic acetylcholine receptors using rat striatum and whole brain membrane preparations, respectively. This series of compounds exhibited selectivity for α4β2* nAChRs and did not interact w...

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Detalles Bibliográficos
Main Authors: Chen, Jianhong, Norrholm, Seth, Dwoskin, Linda P., Crooks, Peter A., Bai, Donglu
Formato: Artigo
Idioma:Inglês
Publicado: 2003
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Acceso en liña:https://ncbi.nlm.nih.gov/pmc/articles/PMC3749776/
https://ncbi.nlm.nih.gov/pubmed/12467625
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