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Selective targeting of distinct active site nucleophiles by irreversible Src-family kinase inhibitors

Src-family tyrosine kinases play pivotal roles in human physiology and disease, and several drugs that target members of this family are in clinical use. None of these drugs appear to discriminate among closely related kinases. However, assessing their selectivity toward endogenous kinases in living...

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Detalhes bibliográficos
Main Authors: Gushwa, Nathan N., Kang, Sumin, Chen, Jing, Taunton, Jack
Formato: Artigo
Idioma:Inglês
Publicado em: 2012
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC3729023/
https://ncbi.nlm.nih.gov/pubmed/23190395
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/ja310659j
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