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Discriminative stimulus functions in rats of AM1346, a high-affinity CB1R selective anandamide analog

OBJECTIVE: To characterize in vivo the high-affinity CB(1) cannabinoid receptor (CB(1)R) selective anandamide analog AM1346 [alkoxyacid amide of N-eicosa-tetraenylamine] using drug discrimination. Substitution tests involved Δ(9)-tetrahydrocannabinol (Δ(9)-THC) and R-(+)-methanandamide (mAEA), a met...

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Autors principals: Järbe, Torbjörn U. C., Li, Chen, Liu, Qian, Makriyannis, Alexandros
Format: Artigo
Idioma:Inglês
Publicat: 2008
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Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC3727224/
https://ncbi.nlm.nih.gov/pubmed/18521574
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1007/s00213-008-1199-3
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