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Drug Promiscuity in PDB: Protein Binding Site Similarity Is Key

Drug repositioning applies established drugs to new disease indications with increasing success. A pre-requisite for drug repurposing is drug promiscuity (polypharmacology) – a drug’s ability to bind to several targets. There is a long standing debate on the reasons for drug promiscuity. Based on la...

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Autors principals: Haupt, V. Joachim, Daminelli, Simone, Schroeder, Michael
Format: Artigo
Idioma:Inglês
Publicat: Public Library of Science 2013
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Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC3689763/
https://ncbi.nlm.nih.gov/pubmed/23805191
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1371/journal.pone.0065894
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