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l-Aminoacyl-triazine Derivatives Are Isoform-Selective PI3Kβ Inhibitors That Target Nonconserved Asp862 of PI3Kβ

[Image: see text] A series of aminoacyl-triazine derivatives based upon the pan-PI3K inhibitor ZSTK474 were identified as potent and isoform-selective inhibitors of PI3Kβ. The compounds showed selectivity based upon stereochemistry with l-amino acyl derivatives preferring PI3Kβ, while their d-congen...

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Detalhes bibliográficos
Main Authors: Pinson, Jo-Anne, Zheng, Zhaohua, Miller, Michelle S., Chalmers, David K., Jennings, Ian G., Thompson, Philip E.
Formato: Artigo
Idioma:Inglês
Publicado em: American Chemical Society 2012
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC3688631/
https://ncbi.nlm.nih.gov/pubmed/23795239
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/ml300336j
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