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N-methyl-substituted fluorescent DAG-indololactone isomers exhibit dramatic differences in membrane interactions and biological activity

N-methyl substituted diacylglycerol-indololactones (DAG-indololactones) are newly-synthesized effectors of protein kinase C (PKC) isoforms and exhibit substantial selectivity between RasGRP3 and PKC alpha. We present a comprehensive analysis of membrane interactions and biological activities of seve...

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Detalhes bibliográficos
Main Authors: Gal, Noga, Kolusheva, Sofiya, Kedei, Noemi, Telek, Andrea, Naeem, Taiyabah A., Lewin, Nancy E., Lim, Langston, Mannan, Poonam, Garfield, Susan H., Kazzouli, Säid El, Sigano, Dina M., Marquez, Victor E., Blumberg, Peter M., Jelinek, Raz
Formato: Artigo
Idioma:Inglês
Publicado em: 2011
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Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC3665409/
https://ncbi.nlm.nih.gov/pubmed/23106081
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