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Funnel metadynamics as accurate binding free-energy method

A detailed description of the events ruling ligand/protein interaction and an accurate estimation of the drug affinity to its target is of great help in speeding drug discovery strategies. We have developed a metadynamics-based approach, named funnel metadynamics, that allows the ligand to enhance t...

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Autors principals: Limongelli, Vittorio, Bonomi, Massimiliano, Parrinello, Michele
Format: Artigo
Idioma:Inglês
Publicat: National Academy of Sciences 2013
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Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC3631651/
https://ncbi.nlm.nih.gov/pubmed/23553839
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1073/pnas.1303186110
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