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Discovery of Allosteric Modulators of Factor XIa by Targeting Hydrophobic Domains Adjacent to its Heparin-Binding Site

To discover promising sulfated allosteric modulators (SAMs) of glycosaminoglycan-binding proteins (GBPs), such as human factor XIa (FXIa), we screened a library of 26 synthetic, sulfated quinazolin-4(3H)-ones (QAOs) resulting in the identification of six molecules that reduced the V(MAX) of substrat...

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Autori principali: Karuturi, Rajesh, Al-Horani, Rami A., Mehta, Shrenik C., Gailani, David, Desai, Umesh R.
Natura: Artigo
Lingua:Inglês
Pubblicazione: 2013
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC3625964/
https://ncbi.nlm.nih.gov/pubmed/23451707
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/jm301757v
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