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Fine-Tuning S1P Therapeutics

Sphingosine 1-phosphate receptor-1 (S1P(1)), a novel therapeutic target for multiple sclerosis, regulates lymphocyte trafficking, heart rate, and vascular function. The discovery of NIBR-0213, a competitive antagonist for S1P(1) that inhibits autoimmune inflammation while sparing bradycardia (Quanca...

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Bibliografiske detaljer
Main Authors: Obinata, Hideru, Hla, Timothy
Format: Artigo
Sprog:Inglês
Udgivet: 2012
Fag:
Online adgang:https://ncbi.nlm.nih.gov/pmc/articles/PMC3625427/
https://ncbi.nlm.nih.gov/pubmed/22999874
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.chembiol.2012.09.002
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