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An optimized RAD51 inhibitor that disrupts homologous recombination without requiring Michael acceptor reactivity

Homologous recombination (HR) is an essential process in cells that provides repair of DNA double-strand breaks and lesions that block DNA replication. RAD51 is an evolutionarily conserved protein that is central to HR. Overexpression of RAD51 protein is common in cancer cells and represents a poten...

Deskribapen osoa

Gorde:
Xehetasun bibliografikoak
Egile Nagusiak: Budke, Brian, Kalin, Jay H., Pawlowski, Michal, Zelivianskaia, Anna S., Wu, Megan, Kozikowski, Alan P., Connell, Philip P.
Formatua: Artigo
Hizkuntza:Inglês
Argitaratua: 2012
Gaiak:
Sarrera elektronikoa:https://ncbi.nlm.nih.gov/pmc/articles/PMC3619390/
https://ncbi.nlm.nih.gov/pubmed/23231413
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/jm301565b
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