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Predicting Intrinsic Clearance for Drugs and Drug Candidates Metabolized by Aldehyde Oxidase
Metabolism by aldehyde oxidase (AO) has been responsible for a number of drug failures in clinical trials. The main reason is the clearance values for drugs metabolized by AO are underestimated by allometric scaling from preclinical species. Furthermore, in vitro human data also underestimates clear...
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| Autori principali: | , |
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| Natura: | Artigo |
| Lingua: | Inglês |
| Pubblicazione: |
2013
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| Soggetti: | |
| Accesso online: | https://ncbi.nlm.nih.gov/pmc/articles/PMC3615103/ https://ncbi.nlm.nih.gov/pubmed/23363487 https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/mp300568r |
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