Cargando...

Contribution of OATP1B1 and OATP1B3 to the Disposition of Sorafenib and Sorafenib-Glucuronide

PURPOSE: Many tyrosine kinase inhibitors (TKIs) undergo extensive hepatic metabolism, but mechanisms of their hepatocellular uptake remain poorly understood. We hypothesized that liver uptake of TKIs is mediated by the solute carriers OATP1B1 and OATP1B3. EXPERIMENTAL DESIGN: Transport of crizotinib...

Descrición completa

Gardado en:
Detalles Bibliográficos
Main Authors: Zimmerman, Eric I., Hu, Shuiying, Roberts, Justin L., Gibson, Alice A., Orwick, Shelley J., Li, Lie, Sparreboom, Alex, Baker, Sharyn D.
Formato: Artigo
Idioma:Inglês
Publicado: 2013
Assuntos:
Acceso en liña:https://ncbi.nlm.nih.gov/pmc/articles/PMC3602278/
https://ncbi.nlm.nih.gov/pubmed/23340295
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1158/1078-0432.CCR-12-3306
Tags: Engadir etiqueta
Sen Etiquetas, Sexa o primeiro en etiquetar este rexistro!