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Nanomolar Potency and Metabolically Stable Inhibitors of Kidney Urea Transporter UT-B

Urea transporters, which include UT-B in kidney microvessels, are potential targets for development of drugs with a novel diuretic (‘urearetic’) mechanism. We recently identified, by high-throughput screening, a triazolothienopyrimidine UT-B inhibitor, 1, that selectively and reversibly inhibited ur...

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Autors principals: Anderson, Marc O., Zhang, Jicheng, Liu, Yan, Yao, Chenjuan, Phuan, Puay-Wah, Verkman, A. S.
Format: Artigo
Idioma:Inglês
Publicat: 2012
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC3590912/
https://ncbi.nlm.nih.gov/pubmed/22694147
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/jm300491y
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