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Pyruvate dehydrogenase kinase as a novel therapeutic target in oncology

Current drug development in oncology is non-selective as it typically focuses on pathways essential for the survival of all dividing cells. The unique metabolic profile of cancer, which is characterized by increased glycolysis and suppressed mitochondrial glucose oxidation (GO) provides cancer cells...

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Détails bibliographiques
Auteurs principaux: Sutendra, Gopinath, Michelakis, Evangelos D.
Format: Artigo
Langue:Inglês
Publié: Frontiers Media S.A. 2013
Sujets:
Accès en ligne:https://ncbi.nlm.nih.gov/pmc/articles/PMC3590642/
https://ncbi.nlm.nih.gov/pubmed/23471124
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3389/fonc.2013.00038
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